AMITRIPTYLINE
Strength10 mg
Formoral.solid
10-25 mg once daily at bedtime, titrate by 10-25 mg every 2-4 weeks up to 50-75 mg daily - long-term
Specialist pediatric urology referral
AUA Guideline on Diagnosis and Treatment of Interstitial Cystitis/Bladder Pain Syndrome 2022 for the indication, with the figures from Amitriptyline Hydrochloride 25 mg Film-Coated Tablets SmPC section 4.2 (eMC product 13683): "The initial dose should be 10 mg - 25 mg in the evening. Doses can be increased with 10 mg - 25 mg every 3 - 7 days as tolerated Recommended doses are 25 mg - 75 mg daily in the evening." The 50 mg step is the same section's "Initially 25 mg 2 times daily (50 mg daily)". The SmPC carries no interstitial cystitis indication; that is from the urology guideline, which is not held in this corpus.
Tricyclic antidepressant used at low dose for its central and peripheral pain-modulating and anticholinergic effects rather than as an antidepressant, calming the bladder pain and urgency of interstitial cystitis. First-line oral neuromodulator per AUA guidance.
- Amitriptyline is the first-line oral neuromodulatory medication for bladder pain syndrome.
- Anticholinergic side effects include sedation, dry mouth, and constipation; administer at bedtime.
- Contraindicated in recent myocardial infarction and cardiac arrhythmia.
- Avoid in elderly patients, and in severe cardiovascular disease or arrhythmias. Amitriptyline - StatPearls - NCBI Bookshelf (NBK537225) puts amitriptyline on the American Geriatrics Society's Beers list, to be avoided in the elderly because its anticholinergic effect is so strong.
| Egyptian brand | Manufacturer | Indicative price |
|---|---|---|
| TRYPTIZOL 10 MG 20 TABS. | KAHIRA | 10.00 EGP (0.50/unit) |
| TRYPTIZOL 10 MG 60 TABS. | KAHIRA | 30.00 EGP (0.50/unit) |
| GRANITYLLIN 25MG/5ML SYP. 120 ML? strength differs? different route - not oral solid | GRAND PHARMA > DELTA GRAND PHARMA | 5.00 EGP |
| ZINOTRAVAL 25MG/5ML SYP. 120 ML? strength differs? different route - not oral solid | DEBEIKY > PHARMACHEMIC | 10.00 EGP |