CABERGOLINE
Strength0.5 mg
Formoral.solid
0.5 mg weekly (administered as 0.25 mg twice weekly), titrate by 0.5 mg/week monthly up to max 4.5 mg/week based on prolactin levels - long-term
Specialist pediatric endocrinology management
Endocrine Society Guideline on Pituitary Tumors 2011
Dopamine agonist that suppresses prolactin secretion by stimulating pituitary D2 receptors; first-line therapy for hyperprolactinaemia given its efficacy and tolerability advantage over bromocriptine, started only after pregnancy, hypothyroidism, and drug-induced causes have been excluded.
- Cabergoline is the first-line dopamine agonist, with superior efficacy and tolerability over bromocriptine.
- Exclude pregnancy, hypothyroidism, and drug-induced causes (antipsychotics, metoclopramide) before starting.
- Perform baseline echocardiogram if high doses (>2 mg/week) or prolonged high-dose therapy are used due to risk of cardiac valvulopathy.
| Egyptian brand | Manufacturer | Indicative price |
|---|---|---|
| CABERGOLACTO 0.5 MG 2 TABS. | IDI > NOVELL PHARMA | 36.00 EGP (18.00/unit) |
| CABERGLOBE 0.5 MG 2 TABS. | EGPI > GLOBE INTERNATIONAL PHARMACEUTICALS | 45.00 EGP (22.50/unit) |
| MARVIGOLINE 0.5 MG 2 TABS. | RAMEDA | 66.00 EGP (33.00/unit) |
| CABROSTINEX 0.5 MG 8 TABS. | MEDIZEN PHARMACEUTICAL INDUSTRIES > ROTABIOGEN | 339.00 EGP (42.38/unit) |
| GOLINOTECH 0.5 MG 2 TABS. | EUROPEAN EGYPTIAN PHARM. IND. > PHARMA-TECH | 103.00 EGP (51.50/unit) |
| DOSTILACT 0.5 MG 2 TABS. | ATCO PHARMA > OMEGA PHARMA OPCI | 105.00 EGP (52.50/unit) |
| DOSTINEX 0.5 MG 2 TABS. | PFIZER | 172.00 EGP (86.00/unit) |
| DELCABRIN 0.5 MG 2 SCORED TABS. | EGPI > HEALTH WELL EGYPT | 105.00 EGP |